BDBM50157430 CHEMBL3781271

SMILES C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)c1ccc(Br)cc1)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCC[N+](C)(C)C)C(=O)N[C@@H](CO)C(N)=O

InChI Key InChIKey=PBXKOVFJOWCAAC-JGLPLDBMSA-O

Data  4 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50157430   

TargetChromobox protein homolog 7(Homo sapiens (Human))
University Of Victoria

Curated by ChEMBL
LigandPNGBDBM50157430(CHEMBL3781271)
Affinity DataIC50:  1.70E+3nMAssay Description:Binding affinity to N-terminal His6-tagged human CBX7 (8 to 62) expressed in Escherichia coli BL21 using FITC-peptide-3 as competitive binding probe ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChromobox protein homolog 8(Homo sapiens (Human))
University Of Victoria

Curated by ChEMBL
LigandPNGBDBM50157430(CHEMBL3781271)
Affinity DataIC50:  4.20E+4nMAssay Description:Inhibition of CBX8 (unknown origin) assessed as inhibition of CBX4 disruption by competitive FP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChromobox protein homolog 7(Homo sapiens (Human))
University Of Victoria

Curated by ChEMBL
LigandPNGBDBM50157430(CHEMBL3781271)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of CBX7 (unknown origin) assessed as inhibition of CBX4 disruption by competitive FP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChromobox protein homolog 6(Homo sapiens (Human))
University Of Victoria

Curated by ChEMBL
LigandPNGBDBM50157430(CHEMBL3781271)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of CBX6 (unknown origin) assessed as inhibition of CBX4 disruption by competitive FP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed