BDBM50159419 CHEMBL262379::Des-AA1,2,5-[D-Trp8,Tyr11]SRIF

SMILES C[C@@H](O)[C@H]1NC(=O)[C@H](CCCCN)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H](Cc2ccccc2)NC(=O)[C@@H](CCCCN)NC(=O)[C@H](N)CSSC[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](Cc2ccc(O)cc2)NC1=O)[C@@H](C)O)C(O)=O

InChI Key InChIKey=NIVBKEGMFSFLSD-KGVPGVLISA-N

Data  5 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50159419   

TargetSomatostatin receptor type 4(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50159419(CHEMBL262379 | Des-AA1,2,5-[D-Trp8,Tyr11]SRIF)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of [Leu8,D-Trp22,125I-Tyr25]SRIF-28 binding to human somatostatin receptor type 4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50159419(CHEMBL262379 | Des-AA1,2,5-[D-Trp8,Tyr11]SRIF)
Affinity DataIC50:  16nMAssay Description:Inhibition of [Leu8,D-Trp22,125I-Tyr25]SRIF-28 binding to human somatostatin receptor type 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50159419(CHEMBL262379 | Des-AA1,2,5-[D-Trp8,Tyr11]SRIF)
Affinity DataIC50:  8nMAssay Description:Inhibition of [Leu8,D-Trp22,125I-Tyr25]SRIF-28 binding to human somatostatin receptor type 3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50159419(CHEMBL262379 | Des-AA1,2,5-[D-Trp8,Tyr11]SRIF)
Affinity DataIC50:  10nMAssay Description:Inhibition of [Leu8,D-Trp22,125I-Tyr25]SRIF-28 binding to human somatostatin receptor type 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50159419(CHEMBL262379 | Des-AA1,2,5-[D-Trp8,Tyr11]SRIF)
Affinity DataIC50:  4.80nMAssay Description:Inhibition of [Leu8,D-Trp22,125I-Tyr25]SRIF-28 binding to human somatostatin receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed