BDBM50164033 CHEMBL183380::N-[2,2'']Bithiophenyl-5-ylmethyl-N''-(2''-sulfamoyl-biphenyl-4-ylmethyl)-isophthalamide
SMILES NS(=O)(=O)c1ccccc1-c1ccc(CNC(=O)c2cccc(c2)C(=O)NCc2ccc(s2)-c2cccs2)cc1
InChI Key InChIKey=NMONGYGAHGGEGU-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50164033
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataKi: 6.20E+3nMAssay Description:Inhibitory constant against voltage-gated sodium channel Nav1.7 in electrophysiology assays (EP)More data for this Ligand-Target Pair
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 2.90E+3nMAssay Description:In vitro inhibitory concentration against voltage-gated sodium channel Nav1.7 in voltage-ion-probe-reader (VIPR) assayMore data for this Ligand-Target Pair