BDBM50164037 (1R,2R)-3-Methylene-cyclopropane-1,2-dicarboxylic acid 1-[([2,2'']bithiophenyl-5-ylmethyl)-amide] 2-[(2''-sulfamoyl-biphenyl-4-ylmethyl)-amide]::CHEMBL361535

SMILES NS(=O)(=O)c1ccccc1-c1ccc(CNC(=O)[C@@H]2[C@@H](C(=O)NCc3ccc(s3)-c3cccs3)C2=C)cc1

InChI Key InChIKey=ZFWOLLUJIPGNJU-UIOOFZCWSA-N

Data  1 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50164037   

TargetSodium channel protein type 9 subunit alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50164037((1R,2R)-3-Methylene-cyclopropane-1,2-dicarboxylic ...)
Affinity DataKi:  5.70E+3nMAssay Description:Inhibitory constant against voltage-gated sodium channel Nav1.7 in electrophysiology assays (EP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50164037((1R,2R)-3-Methylene-cyclopropane-1,2-dicarboxylic ...)
Affinity DataIC50:  840nMAssay Description:In vitro inhibitory concentration against voltage-gated sodium channel Nav1.7 in voltage-ion-probe-reader (VIPR) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed