BDBM50164774 (2S,5R)-5-Ethyl-4-methyl-piperazine-2-carboxylic acid [(R)-2-(4-tert-butylcarbamoyl-4-cyclohexyl-piperidin-1-yl)-1-(4-fluoro-benzyl)-2-oxo-ethyl]-amide; dihydrochloride::CHEMBL554368
SMILES CC[C@@H]1CN[C@@H](CN1C)C(=O)N[C@H](Cc1ccc(F)cc1)C(=O)N1CCC(CC1)(C1CCCCC1)C(=O)NC(C)(C)C
InChI Key InChIKey=UTVJDBAFZSBXLX-FCEKVYKBSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50164774
Affinity DataEC50: 330nMAssay Description:Concentration of compound at 50% maximum cAMP accumulation mediated by human melanocortin 4 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 2.40E+3nMAssay Description:Concentration of compound at 50% maximum cAMP accumulation mediated by human melanocortin 5 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 46nMAssay Description:Inhibitory concentration to displace [125I]NDP-alpha-MSH from human melanocortin 4 receptor expressed in CHO cells; Control 19 nMMore data for this Ligand-Target Pair