BDBM50166976 CHEMBL3799455
SMILES COc1cc(CCNCCc2ccc(O)c3[nH]c(=O)ccc23)ccc1OCCCc1ccccc1
InChI Key InChIKey=ROTBWFGDDNEYCJ-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 9 hits for monomerid = 50166976
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander University
Curated by ChEMBL
Friedrich-Alexander University
Curated by ChEMBL
Affinity DataKi: 6.30nMAssay Description:Displacement of [3H]CGP12177 from human beta2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 64nMAssay Description:Displacement of [3H]spiperone from human D2L receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 150nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 160nMAssay Description:Displacement of [3H]spiperone from human D2S receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 900nMAssay Description:Displacement of [3H]spiperone from human D4.4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.80E+3nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 17nMAssay Description:Agonist activity at human D2S receptor expressed in HEK293 cells cotransfected with Gqi5 protein assessed as [3H]IP3 accumulation after 120 mins by s...More data for this Ligand-Target Pair
Affinity DataEC50: 240nMAssay Description:Agonist activity at ARMS2-PK-tagged D2S receptor (unknown origin) transfected in HEK293 cells after 5 hrs by beta-arrestin assayMore data for this Ligand-Target Pair