BDBM50167285 CHEMBL3797780
SMILES Cc1c(cnc2[nH]cnc12)-n1c2cn[nH]c2c2cc(F)ccc12
InChI Key InChIKey=RRCNPYRCOUOTDZ-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50167285
Affinity DataEC50: 251nMAssay Description:Inhibition of human MetAP2 in HUVEC cells assessed as accumulation of N-Met 14-3-3gamma after 24 hrs by western blot analysisMore data for this Ligand-Target Pair
Affinity DataIC50: <5.01E+4nMAssay Description:Inhibition of human CYP1A2 expressed in Escherichia coli DH5alphaMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of recombinant full-length human MetAP2 catalytic domain (110 to 478 residues) expressed in baculovirus using Met-AMC as substrate by fluo...More data for this Ligand-Target Pair