BDBM50169467 4-{3-[2-(5-Chloro-1H-indol-3-yl)-ethylsulfanyl]-5-quinolin-2-yl-[1,2,4]triazol-4-yl}-butylamine::CHEMBL189554
SMILES NCCCCn1c(SCCc2c[nH]c3ccc(Cl)cc23)nnc1-c1ccc2ccccc2n1
InChI Key InChIKey=JZSSOKLDWIJDBZ-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50169467
Affinity DataKi: 2.30nMAssay Description:Inhibitory constant against human sst5 receptor at a dose of 10 uMMore data for this Ligand-Target Pair
Affinity DataKi: 5.60nMAssay Description:Inhibitory constant against human sst2 receptor at a dose of 10 uMMore data for this Ligand-Target Pair
Affinity DataEC50: 52nMAssay Description:Inhibition of forskolin-induced cAMP accumulation in CHO-K1 cells expressing human sst5 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 6.30nMAssay Description:Inhibition of forskolin-induced cAMP accumulation in CHO-K1 cells expressing human sst2 receptorMore data for this Ligand-Target Pair