BDBM50172509 CHEMBL197159::Dipropyl-(R)-4,5,6,7-tetrahydro-pyrazolo[1,5-a]pyridin-5-yl-amine

SMILES CCCN(CCC)[C@@H]1CCn2nccc2C1

InChI Key InChIKey=LVAZPFMWSRDRRK-GFCCVEGCSA-N

Data  11 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 11 hits for monomerid = 50172509   

TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50172509(CHEMBL197159 | Dipropyl-(R)-4,5,6,7-tetrahydro-pyr...)
Affinity DataKi:  2.10E+3nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50172509(CHEMBL197159 | Dipropyl-(R)-4,5,6,7-tetrahydro-pyr...)
Affinity DataKi:  2.70E+3nMAssay Description:Binding affinity towards human dopamine receptor 3 expressed in Chinese hamster ovary cells using [3H]spiperone (0.5 nM) as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50172509(CHEMBL197159 | Dipropyl-(R)-4,5,6,7-tetrahydro-pyr...)
Affinity DataKi:  4.30E+3nMAssay Description:Displacement of [3H]7-OH-DPAT from human dopamine D3 receptor expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50172509(CHEMBL197159 | Dipropyl-(R)-4,5,6,7-tetrahydro-pyr...)
Affinity DataKi:  1.30E+4nMAssay Description:Binding affinity towards human dopamine receptor 4.4 expressed in Chinese hamster ovary cells using [3H]spiperone (0.5 nM) as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50172509(CHEMBL197159 | Dipropyl-(R)-4,5,6,7-tetrahydro-pyr...)
Affinity DataKi: >2.00E+4nMAssay Description:Binding affinity towards porcine dopamine receptor 1 against radioligand [3H]-SCH- 23390More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50172509(CHEMBL197159 | Dipropyl-(R)-4,5,6,7-tetrahydro-pyr...)
Affinity DataKi: >2.00E+4nMAssay Description:Binding affinity towards human dopamine receptor 2 (short) expressed in Chinese hamster ovary cells using [3H]spiperone (0.5 nM) as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50172509(CHEMBL197159 | Dipropyl-(R)-4,5,6,7-tetrahydro-pyr...)
Affinity DataKi: >2.00E+4nMAssay Description:Binding affinity towards human dopamine receptor 2 (long) expressed in Chinese hamster ovary cells using [3H]spiperone (0.5 nM) as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50172509(CHEMBL197159 | Dipropyl-(R)-4,5,6,7-tetrahydro-pyr...)
Affinity DataKi:  5.30E+4nMAssay Description:Displacement of [3H]spiperone from human dopamine D2short receptor expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50172509(CHEMBL197159 | Dipropyl-(R)-4,5,6,7-tetrahydro-pyr...)
Affinity DataKi:  5.50E+4nMAssay Description:Displacement of [3H]spiperone from human dopamine D2long receptor expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50172509(CHEMBL197159 | Dipropyl-(R)-4,5,6,7-tetrahydro-pyr...)
Affinity DataKi:  5.70E+4nMAssay Description:Displacement of [3H]7-OH-DPAT from human dopamine D2long receptor expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50172509(CHEMBL197159 | Dipropyl-(R)-4,5,6,7-tetrahydro-pyr...)
Affinity DataKi:  6.80E+4nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in porcine cerebral cortex after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed