BDBM50172512 CHEMBL196928::Dipropyl-(4,5,6,7-tetrahydro-pyrazolo[1,5-a]pyridin-5-yl)-amine

SMILES CCCN(CCC)C1CCn2nccc2C1

InChI Key InChIKey=LVAZPFMWSRDRRK-UHFFFAOYSA-N

Data  9 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 9 hits for monomerid = 50172512   

TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50172512(CHEMBL196928 | Dipropyl-(4,5,6,7-tetrahydro-pyrazo...)
Affinity DataKi:  6.70nMAssay Description:High binding affinity towards human dopamine receptor 3 expressed in Chinese hamster ovary cells using [3H]spiperone (0.5 nM) as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50172512(CHEMBL196928 | Dipropyl-(4,5,6,7-tetrahydro-pyrazo...)
Affinity DataKi:  58nMAssay Description:High binding affinity towards human dopamine receptor 4.4 expressed in Chinese hamster ovary cells using [3H]spiperone (0.5 nM) as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50172512(CHEMBL196928 | Dipropyl-(4,5,6,7-tetrahydro-pyrazo...)
Affinity DataKi:  160nMAssay Description:High binding affinity towards human dopamine receptor 2 (short) expressed in Chinese hamster ovary cells using [3H]spiperone (0.5 nM) as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50172512(CHEMBL196928 | Dipropyl-(4,5,6,7-tetrahydro-pyrazo...)
Affinity DataKi:  200nMAssay Description:Low binding affinity towards human dopamine receptor 3 expressed in Chinese hamster ovary cells using [3H]spiperone (0.5 nM) as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50172512(CHEMBL196928 | Dipropyl-(4,5,6,7-tetrahydro-pyrazo...)
Affinity DataKi:  220nMAssay Description:High binding affinity towards human dopamine receptor 2 (long) expressed in Chinese hamster ovary cells using [3H]spiperone (0.5 nM) as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50172512(CHEMBL196928 | Dipropyl-(4,5,6,7-tetrahydro-pyrazo...)
Affinity DataKi:  1.60E+3nMAssay Description:Low binding affinity towards human dopamine receptor 4.4 expressed in Chinese hamster ovary cells using [3H]spiperone (0.5 nM) as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50172512(CHEMBL196928 | Dipropyl-(4,5,6,7-tetrahydro-pyrazo...)
Affinity DataKi:  8.50E+3nMAssay Description:Low binding affinity towards human dopamine receptor 2 (short) expressed in Chinese hamster ovary cells using [3H]spiperone (0.5 nM) as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50172512(CHEMBL196928 | Dipropyl-(4,5,6,7-tetrahydro-pyrazo...)
Affinity DataKi:  1.80E+4nMAssay Description:Low binding affinity towards human dopamine receptor 2 (long) expressed in Chinese hamster ovary cells using [3H]spiperone (0.5 nM) as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50172512(CHEMBL196928 | Dipropyl-(4,5,6,7-tetrahydro-pyrazo...)
Affinity DataKi: >2.00E+4nMAssay Description:Binding affinity (low) towards porcine dopamine receptor 1 against radioligand [3H]-SCH- 23390More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed