BDBM50177573 4-(4-(2-(mesitylamino)-6-methylpyridin-3-ylsulfonyl)phenoxy)butanenitrile::CHEMBL372996

SMILES Cc1cc(C)c(Nc2nc(C)ccc2S(=O)(=O)c2ccc(OCCCC#N)cc2)c(C)c1

InChI Key InChIKey=FZUYYRODAFUAJO-UHFFFAOYSA-N

Data  1 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50177573   

TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177573(4-(4-(2-(mesitylamino)-6-methylpyridin-3-ylsulfony...)
Affinity DataKi:  635nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed