BDBM50186348 CHEMBL3824019

SMILES CCNC(=O)c1cc(F)c(cc1F)-c1cc2cnn(C3CCN(CC3)C(=O)OC(C)C)c2cn1

InChI Key InChIKey=IHNVRMAMWYNXJX-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50186348   

TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50186348(CHEMBL3824019)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human GPR119 expressed in Flp-In-T-Rex-HEK293 cells assessed as stimulation of cAMP level measured after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50186348(CHEMBL3824019)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human GPR119 expressed in Flp-In-T-Rex-HEK293 cells after 30 mins by cAMP accumulation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed