BDBM50189502 CHEMBL3827832
SMILES CCCCCCCCNc1cc(=O)[nH]c(=O)[nH]1
InChI Key InChIKey=PFSWASUQURIOOR-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 8 hits for monomerid = 50189502
Affinity DataKi: 0.626nMAssay Description:Displacement of [3H]PSB-1584 from recombinant human GPR84 expressed in CHO cell membranes co-expressing beta-arrestin2 measured after 6 hrs by scinti...More data for this Ligand-Target Pair
Affinity DataEC50: 512nMAssay Description:Agonist activity at human Gi1alpha-coupled GPR84 expressed in baculovirus infected Sf9 insect cells assessed as stimulation of [35S]GTPgammaS binding...More data for this Ligand-Target Pair
Affinity DataEC50: 114nMAssay Description:Agonist activity at recombinant human GPR84 expressed in CHO cells assessed as beta-arrestin 2 recruitment measured after 90 mins by beta-galactosida...More data for this Ligand-Target Pair
Affinity DataEC50: 341nMAssay Description:Agonist activity at recombinant human GPR84 stably expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of forskolin-induced cAMP ...More data for this Ligand-Target Pair
Affinity DataEC50: 1.25E+3nMAssay Description:Agonist activity at recombinant human GPR84 stably expressed in HEK293 cells co-expressing Galpha16 assessed as increase in intracellular calcium mob...More data for this Ligand-Target Pair
Affinity DataEC50: 1.75E+3nMAssay Description:Agonist activity at recombinant human GPR84 expressed in HEK293 cells assessed as beta-arrestin 2 recruitment measured after 20 mins by luciferase re...More data for this Ligand-Target Pair
Affinity DataEC50: 17nMAssay Description:Agonist activity at recombinant human GPR84 expressed in CHO cells co-expressing beta-galactosidase/beta-arrestin2 assessed as inhibition of forskoli...More data for this Ligand-Target Pair
Affinity DataEC50: 105nMAssay Description:Agonist activity at recombinant human GPR84 expressed in HEK293 cells co-expressing Gqi5 assessed as increase in myo-[3H]inositol phosphate accumulat...More data for this Ligand-Target Pair