BDBM50191474 CHEMBL3899488
SMILES Cc1ncc2sc(nn12)C(=O)N1CCCC1c1ccccc1
InChI Key InChIKey=CQZLZZDJBYTSDH-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50191474
Affinity DataIC50: 415nMAssay Description:Inhibition of CDK8 in human 7dF3 cells preincubated for 2 hrs followed by beta-oestradiol addition measured after 24 hrs by luciferase reporter gene ...More data for this Ligand-Target Pair
Affinity DataIC50: 77nMAssay Description:Inhibition of Alexa647 tracer binding to full length recombinant human His-tagged CDK8/cyclin C expressed in Baculovirus expression system preincubat...More data for this Ligand-Target Pair