BDBM50193684 CHEMBL384362::N-(2-(2-oxa-5-azabicyclo[2.2.1]heptan-5-yl)quinolin-6-yl)-3-(4-(trifluoromethyl)phenyl)propanamide
SMILES FC(F)(F)c1ccc(CCC(=O)Nc2ccc3nc(ccc3c2)N2CC3CC2CO3)cc1
InChI Key InChIKey=DCTXDZRQZOKNLS-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50193684
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Displacement of 125I-[Phe13,Tyr19]-MCH from human MCH-R1More data for this Ligand-Target Pair
Affinity DataEC50: 70nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing rat MCH-R1More data for this Ligand-Target Pair