BDBM50193910 CHEMBL218102::N-(3-(2-(diethylamino)ethoxy)phenyl)-7-(2,6-dimethylphenyl)-5-methylbenzo[e][1,2,4]triazin-3-amine::US8481536, 370

SMILES CCN(CC)CCOc1cccc(Nc2nnc3cc(cc(C)c3n2)-c2c(C)cccc2C)c1

InChI Key InChIKey=FIHAXQZQWYILHF-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50193910   

TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Targegen

US Patent
LigandPNGBDBM50193910(CHEMBL218102 | N-(3-(2-(diethylamino)ethoxy)phenyl...)
Affinity DataIC50:  10.2nMT: 2°CAssay Description:Testing of inhibition of kinases in vitro using luciferase-based assay from KinaseGlo, Promega Corp.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Targegen

US Patent
LigandPNGBDBM50193910(CHEMBL218102 | N-(3-(2-(diethylamino)ethoxy)phenyl...)
Affinity DataIC50:  10nMAssay Description:Inhibition of SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Targegen

US Patent
LigandPNGBDBM50193910(CHEMBL218102 | N-(3-(2-(diethylamino)ethoxy)phenyl...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant Src kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed