BDBM50195536 CHEMBL3976962

SMILES Nc1nc(cs1)-c1ccc(cc1)-n1c(Cl)cc2[nH]c(=O)n(-c3cccc(c3)C(O)=O)c(=O)c12

InChI Key InChIKey=XJJWJDXENZWLAZ-UHFFFAOYSA-N

Data  1 EC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50195536   

Target5'-AMP-activated protein kinase catalytic subunit alpha-1/subunit beta-1/subunit gamma-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL

LigandBDBM50195536(CHEMBL3976962)Copy SMILESCopy InChI

Affinity DataEC50:  631nMAssay Description:Activation of full length human His/GST-tagged AMPK alpha1/beta1/gamma1 expressed in baculovirus expression system after 1 hr by Z'Lyte assayMore data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaantibodypediaantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
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