BDBM50195711 3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)-2-(((pyrazin-2-yloxy)carbonyl)methyl)phenyl)propanoic acid::CHEMBL223350

SMILES Cc1oc(nc1CCOc1ccc(CCC(O)=O)c(CNC(=O)Oc2cnccn2)c1)-c1ccccc1

InChI Key InChIKey=CASKZOPCCIBBBW-UHFFFAOYSA-N

Data  2 IC50  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50195711   

TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50195711(3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)-2-((...)
Affinity DataIC50:  17nMAssay Description:Displacement of [3H]2-methyl-2-(4-{3-propyl-(5-pyridin-2yl-thiophene-2-sulfonyl)-amino]-pro-pyl}-phenoxy)-propionic acid from human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50195711(3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)-2-((...)
Affinity DataEC50:  7nMAssay Description:Activity at human PPARgamma in CV1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50195711(3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)-2-((...)
Affinity DataIC50:  53nMAssay Description:Displacement of [3H]2-(4-{2-[3-(2,4-difluoro-phenyl)-1-heptyl-ureido]-ethyl}-phenoxy)-2-methyl-butyric acid from hPPARalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50195711(3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)-2-((...)
Affinity DataEC50:  35nMAssay Description:Activity at human PPARalpha in CV1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed