BDBM50200114 CHEMBL3920498
SMILES CC(=O)Nc1ccc(cc1)-n1cc(nn1)-c1ccc2ccccc2c1
InChI Key InChIKey=IIQONODPFXFUHM-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50200114
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 2.86E+4nMAssay Description:Noncompetitive inhibition of OGT (unknown origin) using variable UDP-GlcNAc levels and fixed CKII peptide level by UDP-Glo glycosyltransferase assayMore data for this Ligand-Target Pair
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 5.98E+4nMAssay Description:Noncompetitive inhibition of OGT (unknown origin) using fixed UDP-GlcNAc levels and variable CKII peptide level by UDP-Glo glycosyltransferase assayMore data for this Ligand-Target Pair
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 6.67E+4nMAssay Description:Inhibition of OGT (unknown origin) assessed as reduction in GlcNAc transfer to CKII peptide incubated for 60 mins by HPLC methodMore data for this Ligand-Target Pair
TargetPolypeptide N-acetylgalactosaminyltransferase 2(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 6.96E+5nMAssay Description:Inhibition of ppGalNAcT2 (unknown origin) in presence of OGT, EA2 and UDP-GlcNAc incubated for 25 mins at 37 degCMore data for this Ligand-Target Pair