BDBM50203086 4-((5-bromo-1-methyl-1H-indol-3-yl)methylene)-3-(1,2,3-thiadiazol-5-yl)-1H-pyrazol-5(4H)-one::CHEMBL398436

SMILES Cn1cc(\C=C2/C(=O)NN=C2c2cnns2)c2cc(Br)ccc12

InChI Key InChIKey=YTWDDCKDXYRRKH-WCIBSUBMSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50203086   

TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50203086(4-((5-bromo-1-methyl-1H-indol-3-yl)methylene)-3-(1...)
Affinity DataIC50:  110nMAssay Description:Inhibition of human cytoplasmic VEGFR2 expressed in baculovirus after 15 mins by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed