BDBM50207825 CHEMBL246739::H-Cdp-Gly-Gly-Phe-Leu-OH

SMILES CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@@H](N)Cc1c(C)cc(cc1C)C(N)=O)C(O)=O

InChI Key InChIKey=AYRRYHMNASIQTF-SDHOMARFSA-N

Data  3 KI  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50207825   

TargetDelta-type opioid receptor(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50207825(CHEMBL246739 | H-Cdp-Gly-Gly-Phe-Leu-OH)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]diprenorphine from human cloned delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50207825(CHEMBL246739 | H-Cdp-Gly-Gly-Phe-Leu-OH)
Affinity DataKi:  9.80nMAssay Description:Displacement of [3H]diprenorphine from human cloned mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50207825(CHEMBL246739 | H-Cdp-Gly-Gly-Phe-Leu-OH)
Affinity DataKi:  1.30E+3nMAssay Description:Displacement of [3H]diprenorphine from human cloned kappa opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50207825(CHEMBL246739 | H-Cdp-Gly-Gly-Phe-Leu-OH)
Affinity DataEC50:  180nMAssay Description:Agonist activity at human cloned mu opioid receptor assessed as stimulation of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50207825(CHEMBL246739 | H-Cdp-Gly-Gly-Phe-Leu-OH)
Affinity DataEC50:  4.10nMAssay Description:Agonist activity at human cloned delta opioid receptor assessed as stimulation of [35S]GTP-gamma-S bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed