BDBM50209764 CHEMBL3884776

SMILES O[C@H]1COc2cc(F)c(F)c(Nc3ccc(I)cc3F)c2NS(=O)(=O)C2(CC2)C[C@H]1O

InChI Key InChIKey=FENWEVRRFMFDBS-KGLIPLIRSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50209764   

TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Columbia University

Curated by ChEMBL
LigandPNGBDBM50209764(CHEMBL3884776)
Affinity DataIC50:  21nMAssay Description:Inhibition of full length human GST-tagged MEK1 using ERK1/ERK2 peptide substrate in presence of ATP by ADP-Glo chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed