BDBM50210461 (stilbamidine)4-[2-[4-amino(imino)methylphenyl]-(E)-1-ethenyl]phenyl-iminomethanamine::4,4'-(ethene-1,2-diyl)dibenzimidamide::4-((E)-2-{4-[(Z)-amino(imino)methyl]phenyl}vinyl)benzenecarboximidamide::4-((E)-2-{4-[(Z)-amino(imino)methyl]phenyl}vinyl)benzenecarboximidamide(stilbamidine isethionate)::CHEMBL142304::NSC-35605::stilbamidine

SMILES NC(=N)c1ccc(\C=C\c2ccc(cc2)C(N)=N)cc1

InChI Key InChIKey=MMURVNDSFNJHAM-OWOJBTEDSA-N

Data  2 KI  10 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50210461   

TargetHistone-arginine methyltransferase CARM1(Homo sapiens (Human))
The University Of Georgia

Curated by ChEMBL
LigandPNGBDBM50210461((stilbamidine)4-[2-[4-amino(imino)methylphenyl]-(E...)
Affinity DataIC50:  4.00E+5nMAssay Description:Inhibition of GST-tagged CARM1 (unknown origin) using [3H]SAM and histone H3.1 as substrate at 20 uM after 1 hr by P81 filter binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein arginine N-methyltransferase 6(Homo sapiens (Human))
The University Of Georgia

Curated by ChEMBL
LigandPNGBDBM50210461((stilbamidine)4-[2-[4-amino(imino)methylphenyl]-(E...)
Affinity DataIC50:  1.73E+5nMAssay Description:Inhibition of His6x-tagged PRMT6 (unknown origin) using [3H]SAM and histone H3.1 as substrate at 20 uM after 1 hr by P81 filter binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
The University Of Georgia

Curated by ChEMBL
LigandPNGBDBM50210461((stilbamidine)4-[2-[4-amino(imino)methylphenyl]-(E...)
Affinity DataIC50:  4.41E+4nMAssay Description:Inhibition of HA-tagged recombinant PRMT5 (unknown origin) expressed in HEK293T cells using [3H]SAM and histone H4 (1 to 20) as substrate after 8 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
The University Of Georgia

Curated by ChEMBL
LigandPNGBDBM50210461((stilbamidine)4-[2-[4-amino(imino)methylphenyl]-(E...)
Affinity DataIC50:  1.52E+4nMAssay Description:Inhibition of His6x-tagged recombinant PRMT1 (unknown origin) expressed in Escherichia coli BL21(DE3) using [3H]SAM and histone H4 (1 to 20) as subst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed