BDBM50210818 CHEMBL3937015
SMILES O[C@H]1CC[C@@H](CC1)Nc1ncc(-c2ccc3ccccc3c2)c(n1)-c1ccccc1
InChI Key InChIKey=ZQDPBVRIRZFYKQ-YHBQERECSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 50210818
Affinity DataKi: 7.70nMAssay Description:Displacement of [3H]DPCPX from recombinant human adenosine A1 receptor expressed in CHO cell membranes after 1 hr by beta scintillation counting meth...More data for this Ligand-Target Pair
Affinity DataKi: 7.70nMAssay Description:Displacement of [3H]DPCPX from A1 adenosine receptor (unknown origin) expressed in CHO cell membrane incubated for 60 mins at room temperature by NXT...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De Santiago De Compostela
Curated by ChEMBL
Universidade De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 1.37E+3nMAssay Description:Displacement of [3H]SCH-58261 from A2A adenosine receptor (unknown origin) expressed in HEK cell membrane incubated for 60 mins at room temperature b...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De Santiago De Compostela
Curated by ChEMBL
Universidade De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 1.39E+3nMAssay Description:Displacement of [3H]ZM241385 from recombinant human adenosine A2A receptor expressed in HEK293 cell membranes after 2 hrs by beta scintillation count...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]PSB603 from recombinant human adenosine A2B receptor expressed in HEK293 cell membranes after 1 hr by beta scintillation counting...More data for this Ligand-Target Pair
Affinity DataEC50: 166nMAssay Description:Inverse agonist activity at recombinant human adenosine A1 receptor expressed in CHO cell membranes assessed as stimulation of [35S]GTPgammaS binding...More data for this Ligand-Target Pair