BDBM50211535 CHEMBL387993::N-((3S,4R)-6-((S)-2-((2,6-dimethylphenylamino)methyl)pyrrolidine-1-carbonyl)-3-hydroxy-2,2-dimethyl-3,4-dihydro-2H-chromen-4-yl)-4-ethylbenzenesulfonamide::rac-trans-N-(6-((S)-2-((2,6-dimethylphenylamino)methyl)pyrrolidine-1-carbonyl)-3-hydroxy-2,2-dimethyl-3,4-dihydro-2H-chromen-4-yl)-4-ethylbenzenesulfonamide
SMILES CCc1ccc(cc1)S(=O)(=O)N[C@H]1[C@H](O)C(C)(C)Oc2ccc(cc12)C(=O)N1CCC[C@H]1CNc1c(C)cccc1C
InChI Key InChIKey=ZGNURVKJDROBKC-RVQNBHMFSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50211535
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Inhibition of human Kv1.5 channel expressed in mouse L929 cells assessed as blockade of ultra rapidly activating potassium current by volatge clamp t...More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of human Kv1.5 channel expressed in mouse L929 cellsMore data for this Ligand-Target Pair