BDBM50214808 CHEMBL320141::GR-199114X

SMILES Fc1ccc(NC(=O)N[C@H]2C(=O)N(CC(=O)N3CCCC3)c3ccccc3N(C3CCCCC3)C2=O)cc1

InChI Key InChIKey=URMOKEJAUAGZGV-VWLOTQADSA-N

Data  2 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50214808   

TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50214808(CHEMBL320141 | GR-199114X)
Affinity DataKi:  2.5nMAssay Description:Tested for its selectivity against human Cholecystokinin type B receptor isolated from a human temporal cortex cDNA library and stably transfected in...More data for this Ligand-Target Pair
In DepthDetails
TargetCholecystokinin receptor type A(Homo sapiens (Human))TBA
LigandPNGBDBM50214808(CHEMBL320141 | GR-199114X)
Affinity DataKi:  79nMAssay Description:Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to the endothelin A receptor of rat aorta membranesMore data for this Ligand-Target Pair
In DepthDetails