BDBM50220688 (R)-N-((S)-1-(4-(tert-butylcarbamoyl)-4-(4,4-dimethylcyclohexyl)piperidin-1-yl)-3-(4-fluorophenyl)-1-oxopropan-2-yl)-4-methylpiperazine-2-carboxamide::CHEMBL249322
SMILES CN1CCN[C@H](C1)C(=O)N[C@@H](Cc1ccc(F)cc1)C(=O)N1CCC(CC1)(C1CCC(C)(C)CC1)C(=O)NC(C)(C)C
InChI Key InChIKey=LNCCYFHBELRZJF-RRPNLBNLSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50220688
Affinity DataIC50: 162nMAssay Description:Binding affinity to human MC4RMore data for this Ligand-Target Pair
Affinity DataEC50: 546nMAssay Description:Antagonist activity at human MC4R assessed as stimulation of cAMP productionMore data for this Ligand-Target Pair
Affinity DataEC50: 1.12E+3nMAssay Description:Antagonist activity at human MC5R assessed as stimulation of cAMP productionMore data for this Ligand-Target Pair
Affinity DataEC50: 241nMAssay Description:Antagonist activity at human MC3R assessed as stimulation of cAMP productionMore data for this Ligand-Target Pair