BDBM50220711 (R)-N-((S)-3-(4-chlorophenyl)-1-(4-(cyanomethyl)-4-cyclopentylpiperidin-1-yl)-1-oxopropan-2-yl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide::CHEMBL248893
SMILES Clc1ccc(C[C@H](NC(=O)[C@H]2Cc3ccccc3CN2)C(=O)N2CCC(CC#N)(CC2)C2CCCC2)cc1
InChI Key InChIKey=INUXQJJHMOGPLU-IZLXSDGUSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50220711
Affinity DataEC50: 196nMAssay Description:Antagonist activity at human MC4R assessed as stimulation of cAMP productionMore data for this Ligand-Target Pair
Affinity DataEC50: 630nMAssay Description:Antagonist activity at human MC5R assessed as stimulation of cAMP productionMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Binding affinity to human MC4RMore data for this Ligand-Target Pair