BDBM50227844 CHEMBL268768
SMILES COc1cc2nc(nc(N)c2cc1OC)N1CCN(CC1)C(=O)\C=C\c1ccccc1
InChI Key InChIKey=IKWCRLCFRBNCER-CMDGGOBGSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50227844
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
National Institute On Aging/Grc
Curated by ChEMBL
National Institute On Aging/Grc
Curated by ChEMBL
Affinity DataIC50: 0.692nMAssay Description:Displacement of [3H]prazosin binding to Alpha-1 adrenergic receptor sites on rat cerebral cortical membranes at 100 nM concentrationMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
National Institute On Aging/Grc
Curated by ChEMBL
National Institute On Aging/Grc
Curated by ChEMBL
Affinity DataKd: 0.412nMAssay Description:Compound is evaluated for receptor binding affinity using 100 nM concentration on rat cerebral cortical membranesMore data for this Ligand-Target Pair