BDBM50232152 (1-(4-fluorophenethyl)piperidin-4-yl)(3-(2-fluoroethoxy)-2-methoxyphenyl)methanol::(3-(2-Fluoroethoxy)-2-methoxyphenyl)-(1-(2-p-fluorophenylethyl)-piperidine-4-yl)-methanol::CHEMBL402143
SMILES COc1c(OCCF)cccc1C(O)C1CCN(CCc2ccc(F)cc2)CC1
InChI Key InChIKey=QCFZUTYIUYQTPW-UHFFFAOYSA-N
Data 25 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 25 hits for monomerid = 50232152
Affinity DataKi: 9nMAssay Description:Displacement of [3H]MDL from rat 5HT2A receptor expressed in GF62 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 9.02nMAssay Description:Displacement of [3H]MDL from rat 5HT2A receptor expressed in GF62 cells by liquid scintillation analyserMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz
Curated by ChEMBL
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz
Curated by ChEMBL
Affinity DataKi: 71nMAssay Description:Inhibition of human cloned 5-HT2C receptor by competitive binding experimentMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz
Curated by ChEMBL
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz
Curated by ChEMBL
Affinity DataKi: 116nMAssay Description:Inhibition of human cloned 5HT7 receptor by competitive binding experimentMore data for this Ligand-Target Pair
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz
Curated by ChEMBL
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz
Curated by ChEMBL
Affinity DataKi: 148nMAssay Description:Inhibition of human cloned alpha2C adrenergic receptor by competitive binding experimentMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz
Curated by ChEMBL
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz
Curated by ChEMBL
Affinity DataKi: 299nMAssay Description:Inhibition of human cloned 5HT2B receptor by competitive binding experimentMore data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz
Curated by ChEMBL
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz
Curated by ChEMBL
Affinity DataKi: 325nMAssay Description:Inhibition of human cloned alpha1B adrenergic receptor by competitive binding experimentMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz
Curated by ChEMBL
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz
Curated by ChEMBL
Affinity DataKi: 374nMAssay Description:Inhibition of human cloned histamine H1 receptor by competitive binding experimentMore data for this Ligand-Target Pair
TargetD(4) dopamine receptor(Homo sapiens (Human))
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz
Curated by ChEMBL
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz
Curated by ChEMBL
Affinity DataKi: 544nMAssay Description:Inhibition of human cloned dopamine D4 receptor by competitive binding experimentMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz
Curated by ChEMBL
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz
Curated by ChEMBL
Affinity DataKi: 706nMAssay Description:Inhibition of human cloned 5HT1D receptor by competitive binding experimentMore data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz
Curated by ChEMBL
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz
Curated by ChEMBL
Affinity DataKi: 899nMAssay Description:Inhibition of human cloned dopamine D1 receptor by competitive binding experimentMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz
Curated by ChEMBL
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz
Curated by ChEMBL
Affinity DataKi: 1.85E+3nMAssay Description:Inhibition of human cloned 5HT1B receptor by competitive binding experimentMore data for this Ligand-Target Pair
TargetHistamine H2 receptor(Homo sapiens (Human))
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz
Curated by ChEMBL
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz
Curated by ChEMBL
Affinity DataKi: 3.18E+3nMAssay Description:Inhibition of human cloned histamine H2 receptor by competitive binding experimentMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz
Curated by ChEMBL
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz
Curated by ChEMBL
Affinity DataKi: 3.52E+3nMAssay Description:Inhibition of human cloned SERT by competitive binding experimentMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz
Curated by ChEMBL
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz
Curated by ChEMBL
Affinity DataKi: 3.89E+3nMAssay Description:Inhibition of human cloned 5HT6 receptor by competitive binding experimentMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz
Curated by ChEMBL
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human cloned 5HT1A receptor by competitive binding experimentMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz
Curated by ChEMBL
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human cloned mu opioid receptor by competitive binding experimentMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz
Curated by ChEMBL
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human cloned 5HT1E receptor by competitive binding experimentMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz
Curated by ChEMBL
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human cloned DAT by competitive binding experimentMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz
Curated by ChEMBL
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human cloned dopamine D2 receptor by competitive binding experimentMore data for this Ligand-Target Pair
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz
Curated by ChEMBL
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human cloned beta3 adrenergic receptor by competitive binding experimentMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz
Curated by ChEMBL
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human cloned alpha2A adrenergic receptor by competitive binding experimentMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz
Curated by ChEMBL
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human cloned 5HT5A receptor by competitive binding experimentMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz
Curated by ChEMBL
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human cloned histamine H3 receptor by competitive binding experimentMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz
Curated by ChEMBL
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human cloned 5HT3 receptor by competitive binding experimentMore data for this Ligand-Target Pair