BDBM50232770 (S)-2-Amino-N-{[(S)-1-((R)-1-carbamoyl-2-naphthalen-2-yl-ethylcarbamoyl)-2-phenyl-ethylcarbamoyl]-methyl}-3-(4-hydroxy-2,6-dimethyl-phenyl)-N-methyl-propionamide::CHEMBL254927::Dmt-Sar-Phe-D-2-Nal-NH

SMILES CN(CC(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](Cc1ccc2ccccc2c1)C(N)=O)C(=O)[C@@H](N)Cc1c(C)cc(O)cc1C

InChI Key InChIKey=LCSGBFCHAFMKLD-QAXCHELISA-N

Data  2 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50232770   

TargetDelta-type opioid receptor(Homo sapiens (Human))
Medical University Of Lodz

Curated by ChEMBL
LigandPNGBDBM50232770((S)-2-Amino-N-{[(S)-1-((R)-1-carbamoyl-2-naphthale...)
Affinity DataEC50: >1.00E+3nMAssay Description:Antagonist activity at delta opioid receptor expressed in CHO cells assessed as release of intracellular calcium ions by aequorin luminescence-based ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Medical University Of Lodz

Curated by ChEMBL
LigandPNGBDBM50232770((S)-2-Amino-N-{[(S)-1-((R)-1-carbamoyl-2-naphthale...)
Affinity DataIC50:  0.0100nMAssay Description:Displacement of [3H]naloxone from mu opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Medical University Of Lodz

Curated by ChEMBL
LigandPNGBDBM50232770((S)-2-Amino-N-{[(S)-1-((R)-1-carbamoyl-2-naphthale...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]naltrindole from delta opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed