BDBM50232770 (S)-2-Amino-N-{[(S)-1-((R)-1-carbamoyl-2-naphthalen-2-yl-ethylcarbamoyl)-2-phenyl-ethylcarbamoyl]-methyl}-3-(4-hydroxy-2,6-dimethyl-phenyl)-N-methyl-propionamide::CHEMBL254927::Dmt-Sar-Phe-D-2-Nal-NH
SMILES CN(CC(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](Cc1ccc2ccccc2c1)C(N)=O)C(=O)[C@@H](N)Cc1c(C)cc(O)cc1C
InChI Key InChIKey=LCSGBFCHAFMKLD-QAXCHELISA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50232770
Affinity DataEC50: >1.00E+3nMAssay Description:Antagonist activity at delta opioid receptor expressed in CHO cells assessed as release of intracellular calcium ions by aequorin luminescence-based ...More data for this Ligand-Target Pair
Affinity DataIC50: 0.0100nMAssay Description:Displacement of [3H]naloxone from mu opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Medical University Of Lodz
Curated by ChEMBL
Medical University Of Lodz
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]naltrindole from delta opioid receptor in rat brain membranesMore data for this Ligand-Target Pair