BDBM50233781 (R)-N-(1-((3-benzyl-3H-imidazo[4,5-b]pyridin-2-yl)methylamino)-1-oxo-3-(2-(trifluoromethyl)phenyl)propan-2-yl)-2-(trifluoromethyl)benzamide::CHEMBL400260

SMILES FC(F)(F)c1ccccc1C[C@@H](NC(=O)c1ccccc1C(F)(F)F)C(=O)NCc1nc2cccnc2n1Cc1ccccc1

InChI Key InChIKey=ROVOFYSXQNIDPA-AREMUKBSSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50233781   

TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50233781((R)-N-(1-((3-benzyl-3H-imidazo[4,5-b]pyridin-2-yl)...)
Affinity DataIC50:  232nMAssay Description:Blockade of human Nav1.7 channel expressed in HEK293 cells by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 10 subunit alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50233781((R)-N-(1-((3-benzyl-3H-imidazo[4,5-b]pyridin-2-yl)...)
Affinity DataIC50:  366nMAssay Description:Blockade of human Nav1.8 channel expressed in HEK293 cells by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed