BDBM50237878 2-(1,3-bis(3-(piperidin-1-yl)propyl)imidazolidin-2-ylidene)malononitrile::CHEMBL257391
SMILES N#C\[#6](C#N)=[#6]-1\[#7](-[#6]-[#6]-[#6]-[#7]-2-[#6]-[#6]-[#6]-[#6]-[#6]-2)-[#6]-[#6]-[#7]-1-[#6]-[#6]-[#6]-[#7]-1-[#6]-[#6]-[#6]-[#6]-[#6]-1
InChI Key InChIKey=PZBOEBLXMXAJNX-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50237878
Affinity DataKi: 2.40nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned histamine H3 receptor expressed in monkey COS7 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Binding affinity to histamine H3 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from histamine H3 receptor in rat striatal membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Antagonist activity at histamine H3 receptor in rat forebrain assessed as inhibition of [3H]histamine release from synaptosomesMore data for this Ligand-Target Pair