BDBM50243674 ((3aR,6aR)-6-(4-(2-((R)-2-methylpyrrolidin-1-yl)ethyl)phenyl)-1,3a,4,6a-tetrahydrocyclopenta[c]pyrrol-2(1H)-yl)(tetrahydro-2H-pyran-4-yl)methanone::CHEMBL471555
SMILES C[C@@H]1CCCN1CCc1ccc(cc1)C1=CC[C@H]2CN(C[C@@H]12)C(=O)C1CCOCC1
InChI Key InChIKey=KTVGKRKFCUTGRP-HFRGRHLUSA-N
Data 3 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50243674
Affinity DataKi: 0.700nMAssay Description:Displacement of N-[3H]methylhistamine from histamine H3 receptor in rat cortex membraneMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in CHOK1 cells by [3H]R(-)-alpha-methylhistamine displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Inverse agonist activity at human H3 receptor expressed in CHOK1 cells by GTPgammaS binding assayMore data for this Ligand-Target Pair