BDBM50246035 2,2,2-Trifluoro-1-(5-{3-[(thiophen-2-ylsulfonyl)methyl]-1,2,4-oxadiazol-5-yl}thiophen-2-yl)ethanone::2,2,2-trifluoro-1-(5-(3-((thiophen-2-ylsulfonyl)methyl)-1,2,4-oxadiazol-5-yl)thiophen-2-yl)ethanone::CHEMBL471174
SMILES FC(F)(F)C(=O)c1ccc(s1)-c1nc(CS(=O)(=O)c2cccs2)no1
InChI Key InChIKey=GJBRKLVHIOIDHV-UHFFFAOYSA-N
Data 6 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 50246035
TargetHistone deacetylase 4(Homo sapiens (Human))
Irbm-Merck Research Laboratories Rome
Curated by ChEMBL
Irbm-Merck Research Laboratories Rome
Curated by ChEMBL
Affinity DataIC50: 35nMAssay Description:Inhibition of His-tagged HDAC4 catalytic domain (unknown origin) expressed in Escherichia coliMore data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
Irbm-Merck Research Laboratories Rome
Curated by ChEMBL
Irbm-Merck Research Laboratories Rome
Curated by ChEMBL
Affinity DataIC50: 520nMAssay Description:Inhibition of HDAC6 (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
Irbm-Merck Research Laboratories Rome
Curated by ChEMBL
Irbm-Merck Research Laboratories Rome
Curated by ChEMBL
TargetHistone deacetylase 3(Homo sapiens (Human))
Irbm-Merck Research Laboratories Rome
Curated by ChEMBL
Irbm-Merck Research Laboratories Rome
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of HDAC3 (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of HDAC1More data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Affinity DataIC50: 3.89E+3nMAssay Description:Inhibition of HDAC1 (unknown origin)More data for this Ligand-Target Pair