BDBM50248427 1,1,1-trifluoro-2-(4-((R)-2-methyl-4-(2-(pyridin-3-yl)ethyl)piperazin-1-ylsulfonyl)phenyl)propan-2-ol::CHEMBL523444
SMILES C[C@@H]1CN(CCc2cccnc2)CCN1S(=O)(=O)c1ccc(cc1)C(C)(O)C(F)(F)F
InChI Key InChIKey=CHXVGBDXNRZKOE-QRIPLOBPSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50248427
Affinity DataIC50: 1.30nMAssay Description:Inhibition of full length human recombinant 11beta-HSD1 expressed in baculovirus insect cell system assessed as conversion of [3H]cortisone to [3H]co...More data for this Ligand-Target Pair
Affinity DataIC50: 29nMAssay Description:Inhibition of full length human recombinant 11beta-HSD1 expressed in HEK293 cells in absence of NADPHMore data for this Ligand-Target Pair