BDBM50250188 4-(5-(4-Chlorophenyl)-3-(cyclopropanecarbonyl)-2-methyl-1H-pyrrol-1-yl)benzenesulfonamide::CHEMBL450053

SMILES Cc1c(cc(-c2ccc(Cl)cc2)n1-c1ccc(cc1)S(N)(=O)=O)C(=O)C1CC1

InChI Key InChIKey=NHOFBVBSHPEQHP-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50250188   

TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50250188(4-(5-(4-Chlorophenyl)-3-(cyclopropanecarbonyl)-2-m...)
Affinity DataEC50:  4.90E+3nMAssay Description:Allosteric modulator activity at alpha7 nAChR in human IMR32 cells assessed as stimulation of agonist-induced intracellular calcium level by FLIPR as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed