BDBM50252868 CHEMBL4081430

SMILES Brc1ccc(CN(c2ccc(Oc3ccccc3)cc2)S(=O)(=O)c2ccc(cc2)C#N)cc1

InChI Key InChIKey=IBYTXPXIACXJSM-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50252868   

TargetGlucocorticoid receptor(Homo sapiens (Human))
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50252868(CHEMBL4081430)
Affinity DataIC50:  7.87E+3nMAssay Description:Antagonist activity at human GRalpha expressed in HEK293 cells assessed as inhibition of dexamethasone-induced response after 24 hrs by luciferase re...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed