BDBM50262508 3-(4-(3-(2-chloro-4-fluorophenyl)-1,2,4-oxadiazol-5-yl)piperidin-1-yl)quinoline::CHEMBL478203

SMILES Fc1ccc(-c2noc(n2)C2CCN(CC2)c2cnc3ccccc3c2)c(Cl)c1

InChI Key InChIKey=YKKVBHCDPMQIEG-UHFFFAOYSA-N

Data  4 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50262508   

TargetCannabinoid receptor 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50262508(3-(4-(3-(2-chloro-4-fluorophenyl)-1,2,4-oxadiazol-...)
Affinity DataEC50:  3.03E+3nMAssay Description:Agonist activity at human CB1 receptor expressed in insect Sf9 cells assessed as effect on Eu-GTP bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50262508(3-(4-(3-(2-chloro-4-fluorophenyl)-1,2,4-oxadiazol-...)
Affinity DataEC50:  89nMAssay Description:Agonist activity at human CB2 receptor expressed in insect Sf9 cells assessed as effect on Eu-GTP bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50262508(3-(4-(3-(2-chloro-4-fluorophenyl)-1,2,4-oxadiazol-...)
Affinity DataEC50:  17nMAssay Description:Agonist activity at human CB2 receptor assessed as inhibition of forskolin-induced increase in intracellular cAMPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50262508(3-(4-(3-(2-chloro-4-fluorophenyl)-1,2,4-oxadiazol-...)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human CB1 receptor assessed as inhibition of forskolin-induced increase in intracellular cAMPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed