BDBM50269950 CHEMBL4100932
SMILES Cl.NCCCCN1N=C(\C=C\c2ccc(O)cc2)c2ccccc2N(Cc2ccc(cc2)-c2ccccc2)C1=O
InChI Key InChIKey=BYQFMPURZVLEPO-LTGZKZEYSA-N
Data 6 EC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 50269950
Affinity DataEC50: 17nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in human urotensin-2-mediated aortic ring contr...More data for this Ligand-Target Pair
Affinity DataEC50: 9.30nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
Affinity DataEC50: 2.19E+3nMAssay Description:Allosteric modulation of human urotensin-2 receptor expressed in HEK293 cells assessed as change in human urotensin-2-induced G12 activation by measu...More data for this Ligand-Target Pair
Affinity DataEC50: 14nMAssay Description:Allosteric modulation of human urotensin-2 receptor expressed in HEK293 cells assessed as change in human urotensin-2-induced Gq activation by measur...More data for this Ligand-Target Pair
Affinity DataEC50: 4.20nMAssay Description:Allosteric modulation of human urotensin-2 receptor expressed in HEK293 cells assessed as change in URP-induced Gq activation by measuring URP pEC50 ...More data for this Ligand-Target Pair
Affinity DataEC50: 117nMAssay Description:Allosteric modulation of human urotensin-2 receptor expressed in HEK293 cells assessed as change in URP-induced G12 activation by measuring URP pEC50...More data for this Ligand-Target Pair