BDBM50275212 CHEMBL4127473

SMILES [#6]-[#6]-[#6](=O)[Se;v2][#6]-[#6](-[#6]-c1cnc(-[#7])c(Cl)c1)-[#6](-[#8])=O

InChI Key InChIKey=DMSZKGIZIIXNLW-UHFFFAOYSA-N

Data  6 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50275212   

TargetCarboxypeptidase N catalytic chain(Homo sapiens (Human))
Showa Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50275212(CHEMBL4127473)
Affinity DataIC50: >3.80E+5nMAssay Description:Inhibition of human carboxypeptidase N preincubated for 10 mins followed by hippuryl-lysine substrate addition measured after 30 mins in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Showa Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50275212(CHEMBL4127473)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of human plasma activated thrombin-activatable fibrinolysis inhibitor after 10 mins in presence of DTTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Showa Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50275212(CHEMBL4127473)
Affinity DataIC50:  3.70E+5nMAssay Description:Inhibition of human plasma activated thrombin-activatable fibrinolysis inhibitor after 10 mins in absence of DTTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B(Sus scrofa)
Showa Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50275212(CHEMBL4127473)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of porcine pancreas carboxypeptidase B after 10 mins in absence of DTTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B(Sus scrofa)
Showa Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50275212(CHEMBL4127473)
Affinity DataIC50:  29nMAssay Description:Inhibition of porcine pancreas carboxypeptidase B after 10 mins in presence of DTTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase N catalytic chain(Homo sapiens (Human))
Showa Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50275212(CHEMBL4127473)
Affinity DataIC50: >3.80E+5nMAssay Description:Inhibition of human carboxypeptidase N preincubated for 10 mins followed by hippuryl-lysine substrate addition measured after 30 mins in absence of D...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed