BDBM50293915 (R)-3,5-Dichloro-4-[6-chloro-4-(1-cyclopropylpropyl)-3-oxo-3,4-dihydropyrazin-2-ylamino]benzonitrile::(R)-3,5-dichloro-4-(6-chloro-4-(1-cyclopropylpropyl)-3-oxo-3,4-dihydropyrazin-2-ylamino)benzonitrile::CHEMBL549538

SMILES CC[C@H](C1CC1)n1cc(Cl)nc(Nc2c(Cl)cc(cc2Cl)C#N)c1=O

InChI Key InChIKey=MQUWREMEXPWUNV-CYBMUJFWSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50293915   

TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50293915((R)-3,5-Dichloro-4-[6-chloro-4-(1-cyclopropylpropy...)
Affinity DataIC50:  1.20nMAssay Description:Displacement of [125I]ovine-CRF from CRF1 receptor in rat frontal cortex by rapid filtration techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50293915((R)-3,5-Dichloro-4-[6-chloro-4-(1-cyclopropylpropy...)
Affinity DataIC50:  1.20nMAssay Description:Displacement of [125I]Tyr-ovine-CRF from CRF1 receptor in rat frontal cortex homogenate by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed