BDBM50293957 5-Chloro-1-(1-ethylpropyl)-3-(2,4,6-trimethylphenylamino)pyrazin-2(1H)-one::CHEMBL570546

SMILES CCC(CC)n1cc(Cl)nc(Nc2c(C)cc(C)cc2C)c1=O

InChI Key InChIKey=LUZPSLKWMMQYTN-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50293957   

TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50293957(5-Chloro-1-(1-ethylpropyl)-3-(2,4,6-trimethylpheny...)
Affinity DataIC50:  2.90nMAssay Description:Displacement of [125I]Tyr-ovine-CRF from CRF1 receptor in rat frontal cortex homogenate by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed