BDBM50294076 4'-((1S,5R)-3-Methyl-3,6-diaza-bicyclo[3.2.0]hept-6-yl)-biphenyl-4-carbonitrile::CHEMBL552506

SMILES CN1C[C@H]2CN([C@H]2C1)c1ccc(cc1)-c1ccc(cc1)C#N

InChI Key InChIKey=PXEWPYFQFZXVIQ-HKUYNNGSSA-N

Data  2 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50294076   

TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50294076(4'-((1S,5R)-3-Methyl-3,6-diaza-bicyclo[3.2.0]hept-...)
Affinity DataKi:  15.9nMAssay Description:Displacement of [3H]N-alpha methyl histamine from human cloned histamine H3 receptor expressed in C6 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50294076(4'-((1S,5R)-3-Methyl-3,6-diaza-bicyclo[3.2.0]hept-...)
Affinity DataKi:  60.3nMAssay Description:Displacement of [3H]N-alpha methyl histamine from rat cortical membrane histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed