BDBM50303576 CHEMBL583473::[1-(2-Morpholin-4-ylethyl)-1H-indol-3-yl](3-noradamantane)-methanone

SMILES O=C(c1cn(CCN2CCOCC2)c2ccccc12)C12CC3CC1CC(C2)C3

InChI Key InChIKey=FLEORYUEILNRHW-UHFFFAOYSA-N

Data  2 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50303576   

TargetCannabinoid receptor 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50303576(CHEMBL583473 | [1-(2-Morpholin-4-ylethyl)-1H-indol...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50303576(CHEMBL583473 | [1-(2-Morpholin-4-ylethyl)-1H-indol...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50303576(CHEMBL583473 | [1-(2-Morpholin-4-ylethyl)-1H-indol...)
Affinity DataEC50:  68nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in HEK293 cells coexpressing Galphaq/o5 assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed