BDBM50303778 (S)-N-((1-carbamimidoylpiperidin-4-yl)methyl)-5-guanidino-2-((S)-2-((S)-5-guanidino-2-(2-phenylacetamido)pentanamido)-3-methylbutanamido)pentanamide::CHEMBL568067
SMILES [#6]-[#6](-[#6])-[#6@H](-[#7]-[#6](=O)-[#6@H](-[#6]-[#6]-[#6]\[#7]=[#6](/[#7])-[#7])-[#7]-[#6](=O)-[#6]-c1ccccc1)-[#6](=O)-[#7]-[#6@@H](-[#6]-[#6]-[#6]\[#7]=[#6](/[#7])-[#7])-[#6](=O)-[#7]-[#6]-[#6]-1-[#6]-[#6]-[#7](-[#6]-[#6]-1)-[#6](-[#7])=[#7]
InChI Key InChIKey=LEEIZVYTIHJJNF-GNKBHMEESA-N
Data 9 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 9 hits for monomerid = 50303778
Affinity DataKi: 53nMAssay Description:Inhibition of human furin by fluorescence assayMore data for this Ligand-Target Pair
TargetProprotein convertase subtilisin/kexin type 6(Homo sapiens (Human))
Philipps University Marburg
Curated by ChEMBL
Philipps University Marburg
Curated by ChEMBL
Affinity DataKi: 67nMAssay Description:Inhibition of human PACE4 expressed in Drosophila schneider 2 cells by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Inhibition of human PC1/3 expressed in Drosophila schneider 2 cells by fluorescence assayMore data for this Ligand-Target Pair
TargetProprotein convertase subtilisin/kexin type 5(Homo sapiens (Human))
Philipps University Marburg
Curated by ChEMBL
Philipps University Marburg
Curated by ChEMBL
Affinity DataKi: 173nMAssay Description:Inhibition of human PC5/6 expressed in Drosophila schneider 2 cells by fluorescence assayMore data for this Ligand-Target Pair
TargetProprotein convertase subtilisin/kexin type 7(Homo sapiens (Human))
Philipps University Marburg
Curated by ChEMBL
Philipps University Marburg
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human PC7 expressed in Drosophila schneider 2 cells by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human PC2 expressed in Drosophila schneider 2 cells by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.00E+4nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 1.23E+5nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of plasminMore data for this Ligand-Target Pair