BDBM50304621 (R)-2-(1-(3-(6-chloronaphthalen-2-ylsulfonyl)-2-hydroxypropanoyl)piperidin-4-yl)-5-methyl-1H-imidazo[1,5-c]imidazol-3(2H)-one::2-(1-{(2R)-3-[(6-Chloronaphthalene-2-yl)sulfonyl]-2-hydroxypropanoyl}piperidin-4-yl)-5-methyl-1,2-dihydro-3Himidazo[1,5-c]imidazol::CHEMBL593236

SMILES Cc1ncc2CN(C3CCN(CC3)C(=O)[C@@H](O)CS(=O)(=O)c3ccc4cc(Cl)ccc4c3)C(=O)n12

InChI Key InChIKey=WSDPDXBHHQAFEA-QFIPXVFZSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50304621   

TargetCoagulation factor X(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50304621((R)-2-(1-(3-(6-chloronaphthalen-2-ylsulfonyl)-2-hy...)
Affinity DataIC50:  21nMAssay Description:Inhibition of human factor 10a by para-nitroanilide release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50304621((R)-2-(1-(3-(6-chloronaphthalen-2-ylsulfonyl)-2-hy...)
Affinity DataIC50:  21nMAssay Description:Inhibition of human factor 10a assessed as p-nitroanilide release using S2765 as substrate by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed