BDBM50314766 CHEMBL1093306::trans-N-(2-((R)-1'-((3R,4S)-1-tert-butyl-4-(2,4-difluorophenyl)pyrrolidine-3-carbonyl)-6-chloro-5-methyl-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl)propan-2-yl)acetamide
SMILES CC(=O)NC(C)(C)[C@@H]1CC2(CCN(CC2)C(=O)[C@H]2CN(C[C@@H]2c2ccc(F)cc2F)C(C)(C)C)c2cc(Cl)c(C)cc12
InChI Key InChIKey=KMNARKQYUZICHM-FULLSBAXSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50314766
Affinity DataIC50: 89nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human MC4R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 94nMAssay Description:Agonist activity at human MC4R expressed in CHO cells assessed as stimulation of intracellular cAMP accumulationMore data for this Ligand-Target Pair