BDBM50336592 2-{[(1S,5R,13R,14S,17S)-10-hydroxy-17-methoxy-4-methyl-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-trien-14-yl]amino}acetic acid::CHEMBL1672084
SMILES CO[C@]12CC[C@H](NCC(O)=O)[C@@H]3Oc4c5c(C[C@H]1N(C)CC[C@@]235)ccc4O
InChI Key InChIKey=YHKUQEWICWSOTO-BSCZKGNESA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 8 hits for monomerid = 50336592
Affinity DataKi: 0.890nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain membrane by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.890nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membranes incubated for 45 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Displacement of [3H][Ile5,6]deltorphin II from delta opioid receptor in rat brain membranes incubated for 45 mins by liquid scintillation counting me...More data for this Ligand-Target Pair
Affinity DataKi: 43nMAssay Description:Displacement of [3H]U69,593 from kappa opioid receptor in guinea-pig brain membranes incubated for 30 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 43nMAssay Description:Displacement of [3H][Ile5,6]deltorphin 2 from delta opioid receptor in Sprague-Dawley rat brain membrane by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataEC50: 399nMAssay Description:Agonist activity at human KOR expressed in CHO cell membranes incubated for 60 mins scintillation counting assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.20nMAssay Description:Agonist activity at human MOR expressed in CHO cell membranes incubated for 60 mins scintillation counting assayMore data for this Ligand-Target Pair
Affinity DataEC50: 9.60nMAssay Description:Agonist activity at human DOR expressed in CHO cell membranes incubated for 60 mins scintillation counting assayMore data for this Ligand-Target Pair