BDBM50347179 CHEMBL1797689
SMILES Oc1ccc2C[C@H]3N(CC4CC4)CC[C@@]4(CC(=O)CC[C@@]34O)c2c1
InChI Key InChIKey=JKSUUZMNWGEVRC-VAMGGRTRSA-N
Data 5 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50347179
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University
Curated by ChEMBL
Kitasato University
Curated by ChEMBL
Affinity DataKi: 0.0380nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellum homogenate by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.140nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig forebrain homogenate by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.648nMAssay Description:Displacement of [3H]U-69,593 from human kappa opioid receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.769nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair